
Tuomo Laitinen
Erikoistutkija
Farmasian laitos, Terveystieteiden tiedekunta
tuomo.laitinen@uef.fi | 040 016 5489
Tietokoneavusteisen lääkeainesuunnittelun dosentti
Julkaisut
74 kappaletta-
Altering distribution profile of palbociclib by its prodrugs
Järvinen, Juulia; Montaser, Ahmed B; Adla, Santosh Kumar; Leppänen, Jukka; Lehtonen, Marko; Vellonen, Kati-Sisko; Laitinen, Tuomo; Jalkanen, Aaro; Elmquist, William F; Timonen, Juri; Huttunen, Kristiina M; Rautio, Jarkko. 2023. European journal of pharmaceutical sciences. 2024; 192: -
Synthesis, Structural and Behavioral Studies of Indole Derivatives D2AAK5, D2AAK6 and D2AAK7 as Serotonin 5-HT1A and 5-HT2A Receptor Ligands
Kaczor, Agnieszka A; Kędzierska, Ewa; Wróbel, Tomasz M; Grudzińska, Angelika; Pawlak, Angelika; Laitinen, Tuomo; Bartyzel, Agata. 2023. Molecules. 28: -
Identification of 4‐Anilinoquin(az)oline as a Cell‐Active Protein Kinase Novel 3 (PKN3) Inhibitor Chemotype**
Asquith, Christopher R. M.; Temme, Louisa; East, Michael P.; Laitinen, Tuomo; Pickett, Julie; Kwarcinski, Frank E.; Sinha, Parvathi; Wells, Carrow I.; Johnson, Gary L.; Zutshi, Reena; Drewry, David H.. 2022. Chemmedchem. 17: . e202200161 -
Optimization of the 4-anilinoquin(az)oline scaffold as epidermal growth factor receptor (EGFR) inhibitors for chordoma utilizing a toxicology profiling assay platform
Bieberich, Andrew A; Laitinen, Tuomo; Maffuid, Kaitlyn; Fatig, Raymond O; Torrice, Chad D; Morris, David C; Crona, Daniel J; Asquith, Christopher RM. 2022. Scientific reports. 12: . 12820 -
PKN3: a target in cancer metastasis
Temme, Louisa; Laitinen, Tuomo; Asquith, Christopher RM. 2022. Nature reviews drug discovery. 21: -
Structural Features Affecting the Interactions and Transportability of LAT1-Targeted Phenylalanine Drug Conjugates
Bahrami, Katayun; Järvinen, Juulia; Laitinen, Tuomo; Reinisalo, Mika; Honkakoski, Paavo; Poso, Antti; Huttunen, Kristiina M.; Rautio, Jarkko. 2022. Molecular pharmaceutics. 2023; 20: 206-218 -
Synthesis and evaluation of 1,2,3-dithiazole inhibitors of the nucleocapsid protein of feline immunodeficiency virus (FIV) as a model for HIV infection
Laitinen, Tuomo; Meili, Theres; Koyioni, Maria; Koutentis, Panayiotis A; Poso, Antti; Hofmann-Lehmann, Regina; Asquith, Christopher RM. 2022. Bioorganic and medicinal chemistry. 68: -
WaterMap‐Guided Structure‐Based Virtual Screening for Acetylcholinesterase Inhibitors
Targowska‐Duda, Katarzyna M.; Maj, Maciej; Drączkowski, Piotr; Budzyńska, Barbara; Boguszewska‐Czubara, Anna; Wróbel, Tomasz M.; Laitinen, Tuomo; Kaczmar, Patrycja; Poso, Antti; Kaczor, Agnieszka A.. 2022. Chemmedchem. 17: . e202100721 -
BCKDK: an emerging kinase target for metabolic diseases and cancer
East, Michael P; Laitinen, Tuomo; Asquith, Christopher RM. 2021. Nature reviews drug discovery. 20: 498 -
Docking-Based 3D-QSAR Studies for 1,3,4-oxadiazol-2-one Derivatives as FAAH Inhibitors
Zieba, Agata; Laitinen, Tuomo; Patel, Jayendra Z.; Poso, Antti; Kaczor, Agnieszka A.. 2021. International journal of molecular sciences. 22: 6108