
PAAVO HONKAKOSKI
Professor
Professor in Biopharmacy. Head of the Discipline
Paavo Honkakoski has a long experience in regulation of drug metabolizing enzymes, drug transporters and nuclear receptors and their applications to assess drug ADMET properties. He is involved in the UEF research community “DrugTech” and a participant in the H2020 consortium project EDCMET. He has accumulated ~3 M€ competitive research funding. He has ~115 peer-reviewed papers garnering >5700 citations. He is active in both graduate and PhD education, having supervised >50 MSc and 11 PhD theses. He is a member of several editorial boards in journals related to drug research. He has served as a director of Graduate Schools/Doctoral Programs in drug research (2008-2017) and Vice Dean of the Faculty of Health Sciences at UEF with responsibilities in research infrastructures and doctoral programs (2012-2017).
Contact info
Organization
Faculty of Health Sciences, School of Pharmacy
paavo.honkakoski@uef.fi
Phone
+358 40 355 2490
Keywords
Teaching Activities
Research groups - UEF
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EDCMET
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Genome Center of Eastern Finland
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Metabolism and transport of drugs and xenobiotics
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Ocular Drug Delivery group (ODD)
Links
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LinkedIn Biography and publications at LinkedIn
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Research gate Description at ResearchGate
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Orcid ORCID profile
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Link My bibliography at NCBI PubMed
Publications
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del Amo, Eva M.; Hammid, Anam; Tausch, Melanie; Toropainen, Elisa; Sadeghi, Amir; Valtari, Annika; Puranen, Jooseppi; Reinisalo, Mika; Ruponen, Marika; Urtti, Arto; Sauer, Achim; Honkakoski, Paavo. 2022. Ocular metabolism and distribution of drugs in the rabbit eye: Quantitative assessment after intracameral and intravitreal administrations International journal of pharmaceutics 613: 121361. 2022
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Saran, Chitra; Sundqvist, Louise; Ho, Henry; Niskanen, Jonna; Honkakoski, Paavo; Brouwer, Kim LR. 2022. Novel Bile Acid-dependent Mechanisms of Hepatotoxicity Associated with Tyrosine Kinase Inhibitors Journal of pharmacology and experimental therapeutics 380 2: 114-125. 2022
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Hammid, Anam; Fallon, John K; Lassila, Toni; Salluce, Giulia; Smith, Philip C; Tolonen, Ari; Sauer, Achim; Urtti, Arto; Honkakoski, Paavo. 2021. Carboxylesterase Activities and Protein Expression in Rabbit and Pig Ocular Tissues Molecular pharmaceutics 18 3: 1305-1316. 2021
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Mechanism-Based Experimental Models for the Evaluation of BSEP Inhibition and DILI. Murphy, William A.; Chitra, Saran; Honkakoski, Paavo; Brouwer, Kim L.R. / Transporters and Drug-Metabolizing Enzymes in Drug Toxicity. 2021. 2021
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Murphy, William A.; Beaudoin, James J.; Laitinen, Tuomo; Sjöstedt, Noora; Malinen, Melina M.; Ho, Henry; Swaan, Peter W.; Honkakoski, Paavo; Brouwer, Kim L.R.. 2021. Identification of Key Amino Acids that Impact Organic Solute Transporter Alpha/Beta (OSTα/ß) Molecular pharmacology 100 6: 599-608. 2021
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Huber, Nadine; Korhonen, Sonja; Hoffmann, Dorit; Leskelä, Stina; Rostalski, Hannah; Remes, Anne M.; Honkakoski, Paavo; Solje, Eino; Haapasalo, Annakaisa. 2021. Deficient neurotransmitter systems and synaptic function in frontotemporal lobar degeneration-Insights into disease mechanisms and current therapeutic approaches Molecular psychiatry Published online: 19 November 2021: 1 - 10. 2021
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Küblbeck, Jenni; Niskanen, Jonna; Honkakoski, Paavo. 2020. Metabolism-Disrupting Chemicals and the Constitutive Androstane Receptor CAR Cells 9 10: 2306. 2020
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Küblbeck, Jenni; Vuorio, Taina; Niskanen, Jonna; Fortino, Vittorio; Braeunin, Albert; Abass, Khaled; Rautio, Arja; Hakkola, Jukka; Honkakoski, Paavo; Levonen, Anna-Liisa. 2020. The EDCMET project: Metabolic effects of endocrine disruptors International journal of molecular sciences 21 8: 3021. 2020
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A Reverse Transfection Method for Screening of Nuclear Receptor Activators. Küblbeck, Jenni; Honkakoski, Paavo / Nuclear Receptors. 2019. 2019
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Giantin, M; Küblbeck, J; Zancanella, V; Prantner, V; Sansonetti, F; Schoeniger, A; Tolosi, R; Guerra, G; Da Ros, S; Dacasto, M; Honkakoski, P. 2019. DNA elements for constitutive androstane receptor- and pregnane X receptor-mediated regulation of bovine CYP3A28 gene PLoS ONE 14 3: e0214338. 2019