
TATU PANTSAR
Senior Researcher
Contact info
Organization
Faculty of Health Sciences, School of Pharmacy
tatu.pantsar@uef.fi
Phone
+358 50 388 1062
Research groups - UEF
Publications
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Andreev, Stanislav; Pantsar, Tatu; Tesch, Roberta; Kahlke, Niclas; El-Gokha, Ahmed; Ansideri, Francesco; Grätz, Lukas; Romasco, Jenny; Sita, Giulia; Geibel, Christian; Lämmerhofer, Michael; Tarozzi, Andrea; Knapp, Stefan; Laufer, Stefan A.; Koch, Pierre. 2021. Addressing a Trapped High-Energy Water: Design and Synthesis of Highly Potent Pyrimidoindole-Based Glycogen Synthase Kinase-3ß Inhibitors Journal of medicinal chemistry 2022; 65 2: 1283-1301. 2021
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Mustonen, Enni-Kaisa; Lee, Serene M L; Niess, Hanno; Schwab, Matthias; Pantsar, Tatu; Burk, Oliver. 2021. Identification and characterization of novel splice variants of human farnesoid X receptor Archives of biochemistry and biophysics 705: 108893. 2021
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Salo-Ahen, Outi MH; Alanko, Ida; Bhadane, Rajendra; Bonvin, Alexandre MJJ; Honorato, Rodrigo Vargas; Hossain, Shakhawath; Juffer, André H; Kabedev, Aleksei; Lahtela-Kakkonen, Maija; Larsen, Anders Støttrup; Lescrinier, Eveline; Marimuthu, Parthiban; Mirza, Muhammad Usman; Mustafa, Ghulam; Nunes-Alves, Ariane; Pantsar, Tatu; Saadabadi, Atefeh; Singaravelu, Kalaimathy; Vanmeert, Michiel. 2021. Molecular Dynamics Simulations in Drug Discovery and Pharmaceutical Development Processes 9 1: 71. 2021
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Andreev, Stanislav; Pantsar, Tatu; El-Gokha, Ahmed; Ansideri, Francesco; Kudolo, Mark; Anton, Débora Bublitz; Sita, Giulia; Romasco, Jenny; Geibel, Christian; Lämmerhofer, Michael; Goettert, Márcia Ines; Tarozzi, Andrea; Laufer, Stefan A; Koch, Pierre. 2020. Discovery and Evaluation of Enantiopure 9 H-pyrimido[4,5- b]indoles as Nanomolar GSK-3ß Inhibitors with Improved Metabolic Stabili International journal of molecular sciences 21 21: 7823. 2020
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Kircher, Theresa; Pantsar, Tatu; Oder, Andreas; Peter von Kries, Jens; Juchum, Michael; Pfaffenrot, Bent; Kloevekorn, Philip; Albrecht, Wolfgang; Selig, Roland; Laufer, Stefan. 2020. Design and synthesis of novel fluorescently labeled analogs of vemurafenib targeting MKK4 European journal of medicinal chemistry 2021; 209: 112901. 2020
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Pantsar, Tatu. 2020. KRAS(G12C)-AMG 510 interaction dynamics revealed by all-atom molecular dynamics simulations Scientific reports 10: 11992. 2020
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Pedreira, Julia G B; Nahidino, Philipp; Kudolo, Mark; Pantsar, Tatu; Berger, Benedict-Tilman; Forster, Michael; Knapp, Stefan; Laufer, Stefan; Barreiro, Eliezer J. 2020. Bioisosteric Replacement of Arylamide-Linked Spine Residues with N-Acylhydrazones and Selenophenes as a Design Strategy to Novel Dibenzosuberone Derivatives as Type I 1/2 p38[alpha] MAP Kinase Inhibitors Journal of medicinal chemistry 63 13: 7347-7354. 2020
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Shevchenko, Ekaterina; Poso, Antti; Pantsar, Tatu. 2020. The autoinhibited state of MKK4: Phosphorylation, putative dimerization and R134W mutant studied by molecular dynamics simulations Computational and Structural Biotechnology Journal 18: 2687-2698. 2020
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Pantsar, Tatu. 2019. The current understanding of KRAS protein structure and dynamics Computational and Structural Biotechnology Journal 2020; 18: 189-198. 2019
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Heider, Fabian; Ansideri, Francesco; Tesch, Roberta; Pantsar, Tatu; Haun, Urs; Döring, Eva; Kudolo, Mark; Poso, Antti; Albrecht, Wolfgang; Laufer, Stefan A; Koch, Pierre. 2019. Pyridinylimidazoles as dual glycogen synthase kinase 3β/p38α mitogen-activated protein kinase inhibitors European journal of medicinal chemistry 175: 309-329. 2019