Tatu Pantsar
Senior Researcher
School of Pharmacy, Faculty of Health Sciences
tatu.pantsar@uef.fi | +358 50 388 1062
Research groups
Publications
26/26 items-
In Silico Evaluation of the Thr58-Associated Conserved Water with KRAS Switch-II Pocket Binders
Leini, Renne; Pantsar, Tatu. 2023. Journal of chemical information and modeling. 63: 1490-1505 -
Decisive role of water and protein dynamics in residence time of p38α MAP kinase inhibitors
Pantsar, Tatu; Kaiser, Philipp D; Kudolo, Mark; Forster, Michael; Rothbauer, Ulrich; Laufer, Stefan A. 2022. Nature communications. 13: . 569 -
Discovery and Development of First-in-Class ACKR3/CXCR7 Superagonists for Platelet Degranulation Modulation
Bayrak, Alp; Mohr, Florian; Kolb, Kyra; Szpakowska, Martyna; Shevchenko, Ekaterina; Dicenta, Valerie; Rohlfing, Anne-Katrin; Kudolo, Mark; Pantsar, Tatu; Günther, Marcel; Kaczor, Agnieszka A.; Poso, Antti; Chevigné, Andy; Pillaiyar, Thanigaimalai; Gawaz, Meinrad; Laufer, Stefan A.. 2022. Journal of medicinal chemistry. 65: 13365–13384 -
Discrepancy in interactions and conformational dynamics of pregnane X receptor (PXR) bound to an agonist and a novel competitive
Rashidian, Azam; Mustonen, Enni-Kaisa; Kronenberger, Thales; Schwab, Matthias; Burk, Oliver; Laufer, Stefan A; Pantsar, Tatu. 2022. Computational and Structural Biotechnology Journal. 20: 3004-3018 -
Regulatory spine RS3 residue of protein kinases: a lipophilic bystander or a decisive element in the small-molecule kinase inhibitor binding?
Shevchenko, Ekaterina; Pantsar, Tatu. 2022. Biochemical society transactions. 50: 633-648 -
Target Hopping from Protein Kinases to PXR: Identification of Small-Molecule Protein Kinase Inhibitors as Selective Modulators of Pregnane X Receptor from TüKIC Library
Mustonen, Enni-Kaisa; Pantsar, Tatu; Rashidian, Azam; Reiner, Juliander; Schwab, Matthias; Laufer, Stefan; Burk, Oliver. 2022. Cells. 11: -
Addressing a Trapped High-Energy Water: Design and Synthesis of Highly Potent Pyrimidoindole-Based Glycogen Synthase Kinase-3ß Inhibitors
Andreev, Stanislav; Pantsar, Tatu; Tesch, Roberta; Kahlke, Niclas; El-Gokha, Ahmed; Ansideri, Francesco; Grätz, Lukas; Romasco, Jenny; Sita, Giulia; Geibel, Christian; Lämmerhofer, Michael; Tarozzi, Andrea; Knapp, Stefan; Laufer, Stefan A.; Koch, Pierre. 2021. Journal of medicinal chemistry. 2022; 65: 1283-1301 -
Identification and characterization of novel splice variants of human farnesoid X receptor
Mustonen, Enni-Kaisa; Lee, Serene M L; Niess, Hanno; Schwab, Matthias; Pantsar, Tatu; Burk, Oliver. 2021. Archives of biochemistry and biophysics. 705: 108893 -
Molecular Dynamics Simulations in Drug Discovery and Pharmaceutical Development
Salo-Ahen, Outi MH; Alanko, Ida; Bhadane, Rajendra; Bonvin, Alexandre MJJ; Honorato, Rodrigo Vargas; Hossain, Shakhawath; Juffer, André H; Kabedev, Aleksei; Lahtela-Kakkonen, Maija; Larsen, Anders Støttrup; Lescrinier, Eveline; Marimuthu, Parthiban; Mirza, Muhammad Usman; Mustafa, Ghulam; Nunes-Alves, Ariane; Pantsar, Tatu; Saadabadi, Atefeh; Singaravelu, Kalaimathy; Vanmeert, Michiel. 2021. Processes. 9: 71 -
Bioisosteric Replacement of Arylamide-Linked Spine Residues with N-Acylhydrazones and Selenophenes as a Design Strategy to Novel Dibenzosuberone Derivatives as Type I 1/2 p38[alpha] MAP Kinase Inhibitors
Pedreira, Julia G B; Nahidino, Philipp; Kudolo, Mark; Pantsar, Tatu; Berger, Benedict-Tilman; Forster, Michael; Knapp, Stefan; Laufer, Stefan; Barreiro, Eliezer J. 2020. Journal of medicinal chemistry. 63: 7347-7354